1-Tosyl-2-trifluoroacetylindole as Promising Partner for Synthesis of Fused Fluorinated Heterocycles

Chunikhin, Konstantin S. (2019) 1-Tosyl-2-trifluoroacetylindole as Promising Partner for Synthesis of Fused Fluorinated Heterocycles. Chemical Science International Journal, 26 (4). pp. 1-4. ISSN 2456-706X

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Abstract

We prepared 1-tosyl-2-trifluoroacetylindole - a novel example of an electron-deficient indole with an electrophilic C(3) position. This substance was involved in cyclocondensation with a variety of amidines to propose a new general pathway to 8H-[4,5-b]indolopyrimidines with yield 50-80%. CF3-containing 5H-[3,2-d]indolopyrimidines were unknown before this study.

Item Type: Article
Subjects: Article Paper Librarian > Chemical Science
Depositing User: Unnamed user with email support@article.paperlibrarian.com
Date Deposited: 03 Apr 2023 09:33
Last Modified: 23 Apr 2024 12:15
URI: http://editor.journal7sub.com/id/eprint/546

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